Detail introduction: Triptorelin/Triptorelin Acetate/140194-24-7
English name | Triptorelin |
CAS NO | 140194-24-7 |
Peptide sequence | Pyr-His-Trp-Ser-Tyr-DTrp-Leu-Arg-Pro-Gly-NH2 |
Molecular formula | C64H82N18O13.C2H4O2 |
Molecular weight | 1371.52 |
storage temperature | 2-8℃ |
purity | ≥98% |
Package | 1mg;5mg;10mg;50mg;100mg,1g or according to customer’s detail requirement. |
Product English synonyms | Triptorelin Acetate; Triptorelin Acetate; Decapeptyl-Depot;6-D-Tryptophan Luteinizing HorMone-Releasing Factor (Pig) Acetate |
What is triptorelin?
Triptorelin Acetate is the acetate of Triptorelin. The active ingredient is triptorelin. Triptorelin is a synthetic high-efficiency agonist analogue. The drug was first marketed in Germany in 1986. In order to increase the bioavailability of general drugs, many salts are formed to increase the solubility and then increase the bioavailability. Therefore, the pharmacological effects and adverse reactions of the two are consistent.
The pharmacological effects of Triptorelin Acetate
The active ingredient of triptorelin acetate is an analogue of synthetic gonadotropin releasing hormone. Its structural modification is to replace the sixth L-glycine in the natural molecular structure with a dextrorotatory color Chemicalbook amino acid to make its agonistic effect more effective. It is significant and the plasma half-life is longer. After the injection of the drug, it will initially stimulate the pituitary to release luteinizing hormone and oocyte maturation hormone. When the pituitary gland enters the refractory period after long-term stimulation, the release of gonadotropins will decrease, thus reducing sex steroids to castrated levels. The above effects are reversible.
The main scope of application of Decapeptyl-Depot
Triptorelin acetate is mainly used to treat endometriosis, hormone-dependent prostate cancer, breast cancer, true precocious puberty in children, and can also be used in assisted reproductive technology.
How to buy Triptorelin in the U. S.
Peptide supplier Remetide specializes in the production and sales of peptides in the USA, as well as Professional Drug peptide R&D. Feel free to contact us if you have any questions or inquiries about Triptorelin Acetate Peptide.