Detail introduction: Deslorelin/deslorelin acetate/DESLORELIN(HUMAN)/57773-65-6/82318-06-7
English name | Deslorelin |
CAS NO | 57773-65-6/82318-06-7 |
Peptide sequence | Pyr-His-Trp-Ser-Tyr-DTrp-Leu-Arg-Pro-NHEt |
Molecular formula | C64H83N17O12 |
Molecular weight | 1282.48 |
storage temperature | 2-8℃ |
purity | ≥98% |
Package | 1mg;5mg;10mg;50mg;100mg,1g or according to customer’s detail requirement. |
Product English synonyms | [D-TRP6, DES-GLY10]-LH-RHETHYLAMIDE;deslorelin acetate; DESLORELIN(HUMAN); DES-GLY10,[D-TRP6]-LH-RHETHYLAMIDE |
What is Deslorelin?
Deslorelin is a synthetic analogue of gonadotrophin-releasing hormone (GnRH), which is more potent than the native hormone and is more resistant to proteolysis Parker and Schimmer. Like GnRH, it binds with high affinity to the GnRH receptor on anterior pituitary cells, where it acts as an agonist.
Acutely, it stimulates the secretion of LH and FSH from the anterior pituitary but prolonged, continuous exposure leads to inhibition of secretion by desensitization of the pituitary gonadotropes. As with other GnRH agonists, it has potential therapeutic applications in the treatment of endometriosis, uterine leiomyoma (fibroids), malignant neoplasms, and assisted reproduction protocols. In pharmaceutical peptides, Deslorelin is a peptide product with a very wide range of applications and a very significant effect.
Dissolution suggestion for Desserelin
Sterile Filtered White lyophilized (freeze-dried) powder. The Deslorelin peptide was lyophilized with no additives. It is recommended to reconstitute the lyophilized Deslorelin in sterile 18MΩ-cm H2O not less than 100μg/ml, which can then be further diluted to other aqueous solutions.
Preservation Suggestions for Desserelin
Lyophilized Deslorelin although stable at room temperature for 3 weeks, should be stored desiccated below -18℃. Upon reconstitution, Deslorelin should be stored at 4℃ between 2-7 days and for future use below -18℃. For long-term storage, it is recommended to add a carrier protein (0.1% HSA or BSA). Please prevent freeze-thaw cycles.
How to buy Deslorelin in the U. S.
Remetide Peptide Supplier specializes in the production and sales of peptides in the USA, as well as Professional Drug peptide R&D. Feel free to contact us if you have any questions or inquiries about Peptides.